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Aripiprazole Lauroxil
CAS No. 1259305-29-7
Aripiprazole Lauroxil ( —— )
产品货号. M26609 CAS No. 1259305-29-7
Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 10MG | ￥332 | 有现货 |
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| 25MG | ￥535 | 有现货 |
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| 50MG | ￥786 | 有现货 |
|
| 100MG | ￥1069 | 有现货 |
|
| 200MG | ￥1604 | 有现货 |
|
| 500MG | ￥2705 | 有现货 |
|
| 1G | 获取报价 | 有现货 |
|
生物学信息
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产品名称Aripiprazole Lauroxil
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.
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产品描述Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic. Aripiprazole lauroxil is cleaved by esterases in vivo to N-hydroxymethyl aripiprazole (lauric acid), which is then cleaved to aripiprazole, which is non-toxic.(In Vivo):Intravenous administration of 1.87?mg/ml Aripiprazole lauroxil bioconversion in vivo involves the formation of an intermediate,?N-hydroxymethyl aripiprazole. The?in vitro?data indicates a high bioconversion of aripiprazole lauroxil, thus, the concentration of?N-hydroxymethyl aripiprazole observed in the animals dosed with aripiprazole lauroxil is surprisingly high.
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同义词——
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通路GPCR/G Protein
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靶点Dopamine Receptor
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受体Mycobacterium tuberculosis
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研究领域——
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适应症——
化学信息
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CAS Number1259305-29-7
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分子量660.7
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分子式C36H51Cl2N3O4
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纯度>98% (HPLC)
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溶解度——
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SMILESCCCCCCCCCCCC(=O)OCN1C(=O)CCc2ccc(OCCCCN3CCN(CC3)c3cccc(Cl)c3Cl)cc12
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Korycka-Machala M, et al. Naphthalimides Selectively Inhibit the Activity of Bacterial, Replicative DNA Ligases and Display Bactericidal Effects against Tubercle Bacilli. Molecules. 2017 Jan 17;22(1). pii: E154.
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